Research Mentor(s)

Antos, John M.

Description

Enzymes have become an attractive option for protein modification chemistry due to the remarkable site-specificity they afford. Of particular interest is sortase A from taphylococcus aureus (SrtAaur), which has garnered attention for its ability to install a variety of non-natural modifications to a conserved oligopeptide substrate. In addition to SrtAaur it has become apparent that sortase A homologs exist in other bacterial strains, each of which is potentially a novel catalyst for protein engineering. Previous work has demonstrated that eight representative sortase A homologs exhibit unique specificities for synthetic peptide substrates, capable of identifying characteristic combinations of amino acids in the “sorting motif.” Presented here is a nucleophile profile of the most promiscuous sortase A homolog investigated, that from Streptococcus pneumoniae (SrtApneu). Exhibiting unique specificities, this SrtA variant may enable unique protein modification chemistry.

Document Type

Event

Start Date

19-5-2016 12:00 PM

End Date

19-5-2016 3:00 PM

Department

Chemistry

Genre/Form

student projects; posters

Subjects – Topical (LCSH)

Enzymes--Analysis; Protein engineering

Type

Image

Keywords

Sortase, nucleophile, transpeptidation, ligation, CRF, peptide

Comments

Outstanding Poster Award Recipient

Rights

Copying of this document in whole or in part is allowable only for scholarly purposes. It is understood, however, that any copying or publication of this documentation for commercial purposes, or for financial gain, shall not be allowed without the author's written permission.

Language

English

Format

application/pdf

Included in

Chemistry Commons

Share

COinS
 
May 19th, 12:00 PM May 19th, 3:00 PM

Evaluating Nucleophile and Substrate Specificities of Sortase A Homologs for Orthogonal Reactivity

Enzymes have become an attractive option for protein modification chemistry due to the remarkable site-specificity they afford. Of particular interest is sortase A from taphylococcus aureus (SrtAaur), which has garnered attention for its ability to install a variety of non-natural modifications to a conserved oligopeptide substrate. In addition to SrtAaur it has become apparent that sortase A homologs exist in other bacterial strains, each of which is potentially a novel catalyst for protein engineering. Previous work has demonstrated that eight representative sortase A homologs exhibit unique specificities for synthetic peptide substrates, capable of identifying characteristic combinations of amino acids in the “sorting motif.” Presented here is a nucleophile profile of the most promiscuous sortase A homolog investigated, that from Streptococcus pneumoniae (SrtApneu). Exhibiting unique specificities, this SrtA variant may enable unique protein modification chemistry.

 

To view the content in your browser, please download Adobe Reader or, alternately,
you may Download the file to your hard drive.

NOTE: The latest versions of Adobe Reader do not support viewing PDF files within Firefox on Mac OS and if you are using a modern (Intel) Mac, there is no official plugin for viewing PDF files within the browser window.